GSK5182
Catalog No: 20375
CAS Number: 877387-37-6 (free base)
Purity: 98% Min.
GSK5182 is a specific inverse agonist for estrogen-related receptor γ.
For research use only. We do not sell to patients.
Chemical Information
| Name | GSK5182 |
|---|---|
| Iupac Chemical Name | 4-[(Z)-1-[4-(2-dimethylaminoethoxy)phenyl]-5-hydroxy-2-phenylpent-1-enyl]phenol |
| Synonyms | GSK5182; GSK 5182; GSK-5182. |
| Molecular Formula | C27H31NO3 |
| Molecular Weight | 417.54 |
| Smile | OC1=CC=C(/C(C2=CC=C(OCCN(C)C)C=C2)=C(C3=CC=CC=C3)\CCCO)C=C1 |
| InChiKey | ZVSFNBNLNLXEFQ-RQZHXJHFSA-N |
| InChi | InChI=1S/C27H31NO3/c1-28(2)18-20-31-25-16-12-23(13-17-25)27(22-10-14-24(30)15-11-22)26(9-6-19-29)21-7-4-3-5-8-21/h3-5,7-8,10-17,29-30H,6,9,18-20H2,1-2H3/b27-26- |
| CAS Number | 877387-37-6 (free base) |
| Related CAS |
Ordering Information
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | Solid powder |
|---|---|
| Purity | 98% Min. |
| Storage | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO |
| Handling | |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| HS Code |
Coming soon.
| Targets | |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |
1: Joo J, Wu Z, Lee B, Shon JC, Lee T, Lee IK, Sim T, Kim KH, Kim ND, Kim SH, Liu KH. In vitro metabolism of an estrogen-related receptor γ modulator, GSK5182, by human liver microsomes and recombinant cytochrome P450s. Biopharm Drug Dispos. 2015 Apr;36(3):163-73. doi: 10.1002/bdd.1929. PubMed PMID: 25451157.
Chemical Structure
